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05-22-3838 BQ-788, Sodium Salt - CAS - Calbiochem

Overview

Key Spec Table

Empirical Formula
C₃₄H₅₀N₅O₇Na

Products

Catalogue NumberPackaging Qty/Pack
05223838-1MGCN 塑膠安瓿;塑膠針藥瓶 1 mg
05223838-5MGCN 塑膠安瓿;塑膠針藥瓶 5 mg
Description
OverviewHighly selective ETB-receptor antagonist (IC50 = 1.2 nM).
Catalogue Number05-22-3838
Brand Family Calbiochem®
SynonymsN-cis-2,6-Dimethylpiperidinocarbonyl-L-γ-MeLeu-D-Trp(MeOCO)-D-Nle-OH, Na
References
ReferencesOkada, M., and Nishikibe, M. 2002. Cardiovasc. Drug Reviews 20, 53.
Taniai, H., et al. 2001. Hepatology 33, 894.
Fukuroda, T., et al. 1994. Biochem. Biophys. Res. Commun. 199, 1461.
Ishikawa, K., et al. 1994. Proc. Natl. Acad. Sci. USA 91, 4892.
Product Information
ATP CompetitiveN
FormWhite to off-white lyophilized solid
Hill FormulaC₃₄H₅₀N₅O₇Na
Chemical formulaC₃₄H₅₀N₅O₇Na
ReversibleN
Structure formula ImageStructure formula Image
Quality LevelMQ100
Biological Information
Primary TargetETB-receptor antagonist
Primary Target IC<sub>50</sub>1.2 nM as ETB-receptor antagonist
Purity≥95% by HPLC
Physicochemical Information
Cell permeableN
Storage and Shipping Information
Ship Code Ambient Temperature Only
Toxicity Standard Handling
Storage -20°C
Protect from Moisture Protect from moisture
Do not freeze Ok to freeze
Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). DMSO and Methano:H₂O stock solutions are stable for up to 2 months at -20°C.
Global Trade Item Number
Catalogue Number GTIN
05223838-1MGCN 04055977225051
05223838-5MGCN 04055977225068