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539636 PKCθ Pseudosubstrate Inhibitor, Myristoylated - Calbiochem

The PKCθ Pseudosubstrate Inhibitor, Myristoylated controls the biological activity of PKCθ. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

MSDS (material safety data sheet) or SDS, CoA and CoQ, dossiers, brochures and other available documents.

Synonyms: Myr-LHQRRGAIKQAKVHHVKC-NH₂, Protein Kinase Cθ Pseudosubstrate Inhibitor, Myristoylated

Primary Target: protein kinase Cθ
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539636
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Overview

Replacement Information

Key Spec Table

Empirical Formula
C₁₀₅H₁₈₂N₃₅O₂₂S

Products

Catalogue NumberPackaging Qty/Pack
539636-500UGCN Plastic ampoule 500 μg
Description
OverviewA cell-permeable, reversible, substrate competitive, myristoylated form of the inhibitor of protein kinase Cθ isozyme pseudosubstrate inhibitor (Cat. No. 539634).
Catalogue Number539636
Brand Family Calbiochem®
SynonymsMyr-LHQRRGAIKQAKVHHVKC-NH₂, Protein Kinase Cθ Pseudosubstrate Inhibitor, Myristoylated
References
ReferencesOsada, S., et al. 1992. Mol. Cell Biol. 12, 3930.
Product Information
ATP CompetitiveY
FormLyophilized solid
FormulationSupplied as a trifluoroacetate salt.
Hill FormulaC₁₀₅H₁₈₂N₃₅O₂₂S
Chemical formulaC₁₀₅H₁₈₂N₃₅O₂₂S
Hygroscopic Hygroscopic
ReversibleY
Quality LevelMQ100
Applications
Biological Information
Primary Targetprotein kinase Cθ
Purity≥95% by HPLC
Physicochemical Information
Cell permeableY
Peptide SequenceMyr-Leu-His-Gln-Arg-Arg-Gly-Ala-Ile-Lys-Gln-Ala-Lys-Val-His-His-Val-Lys-Cys-NH₂
Dimensions
Materials Information
Toxicological Information
Safety Information according to GHS
Safety Information
Product Usage Statements
Storage and Shipping Information
Ship Code Ambient Temperature Only
Toxicity Standard Handling
Storage -20°C
Hygroscopic Hygroscopic
Do not freeze Ok to freeze
Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for 6 months at -20°C.
Packaging Information
Transport Information
Supplemental Information
Specifications
Global Trade Item Number
Catalogue Number GTIN
539636-500UGCN 04055977194807

Documentation

PKCθ Pseudosubstrate Inhibitor, Myristoylated - Calbiochem SDS

Title

Safety Data Sheet (SDS) 

PKCθ Pseudosubstrate Inhibitor, Myristoylated - Calbiochem Certificates of Analysis

TitleLot Number
539636

References

Reference overview
Osada, S., et al. 1992. Mol. Cell Biol. 12, 3930.

Citations

Title
  • Mason, J.C., et al. 2004. Journal of Biological Chemistry 279, 41611.
    		•
    Data Sheet

    Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

    Revision05-September-2008 RFH
    SynonymsMyr-LHQRRGAIKQAKVHHVKC-NH₂, Protein Kinase Cθ Pseudosubstrate Inhibitor, Myristoylated
    DescriptionCell-permeable myristoylated protein kinase Cq pseudosubstrate sequence peptide (Cat. No. 539634). Useful for studies of PKCθ function in intact cells. Sold on the basis of peptide content.
    FormLyophilized solid
    FormulationSupplied as a trifluoroacetate salt.
    Chemical formulaC₁₀₅H₁₈₂N₃₅O₂₂S
    Peptide SequenceMyr-Leu-His-Gln-Arg-Arg-Gly-Ala-Ile-Lys-Gln-Ala-Lys-Val-His-His-Val-Lys-Cys-NH₂
    Purity≥95% by HPLC
    SolubilityH₂O (2 mg/ml)
    Storage -20°C
    Hygroscopic
    Do Not Freeze Ok to freeze
    Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for 6 months at -20°C.
    Toxicity Standard Handling
    ReferencesOsada, S., et al. 1992. Mol. Cell Biol. 12, 3930.
    Citation
  • Mason, J.C., et al. 2004. Journal of Biological Chemistry 279, 41611.
    		•