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505894 CGP 7930 - CAS 57717-80-3 - Calbiochem

505894
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Overview

Replacement Information

Key Spec Table

CAS #Empirical Formula
57717-80-3C₁₉H₃₂O₂

Products

Catalogue NumberPackaging Qty/Pack
5.05894.0001 Sklená flaša 10 mg
Description
OverviewA blood brain barrier permeable, positive allosteric modulator of the metabotropic GABAB receptor. Shown to modulate GABAB receptor in the high affinity state and thereby increases agonist affinity for the receptor. Also enhances agonist potency and efficacy even on recombinant GABAB receptors. Exhibits anxiolytic effects in rodents.
Catalogue Number505894
Brand Family Calbiochem®
SynonymsGABA B Receptor Antagonist, CGP7930, CGP 7930, CGP-7930
References
ReferencesAdams, C. et al., 2007. CNS Drug Rev. 13, 308.
Pin, J.P., et al., 2007. Curr. Neuropharmacol. 5, 195.
Product Information
CAS number57717-80-3
FormPale yellow solid
Hill FormulaC₁₉H₃₂O₂
Chemical formulaC₁₉H₃₂O₂
Structure formula ImageStructure formula Image
Quality LevelMQ100
Applications
Biological Information
Primary TargetGABAB
Purity≥98% by HPLC
Physicochemical Information
Dimensions
Materials Information
Toxicological Information
Safety Information according to GHS
Safety Information
Product Usage Statements
Storage and Shipping Information
Ship Code Shipped at Ambient Temperature or with Blue Ice or with Dry Ice
Toxicity Standard Handling
Storage +2°C to +8°C
Protect from Light Protect from light
Do not freeze Ok to freeze
Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
Packaging Information
Transport Information
Supplemental Information
Specifications
Global Trade Item Number
Catalogue Number GTIN
5.05894.0001 04055977262483

Documentation

CGP 7930 - CAS 57717-80-3 - Calbiochem MSDS

Title

Safety Data Sheet (SDS) 

References

Reference overview
Adams, C. et al., 2007. CNS Drug Rev. 13, 308.
Pin, J.P., et al., 2007. Curr. Neuropharmacol. 5, 195.

Brochure

Title
New Products Flyer- Feb 2014 - Vol 1
Data Sheet

Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

Revision20-September-2013 JSW
SynonymsGABA B Receptor Antagonist, CGP7930, CGP 7930, CGP-7930
DescriptionA blood brain barrier permeable, positive allosteric modulator of the metabotropic GABAB receptor. Shown to modulate GABAB receptor in the high affinity state and thereby increases agonist affinity for the receptor. Also enhances agonist potency and efficacy even on recombinant GABAB receptors. Exhibits anxiolytic effects in rodents.
FormPale yellow solid
CAS number57717-80-3
Chemical formulaC₁₉H₃₂O₂
Structure formulaStructure formula
Purity≥98% by HPLC
SolubilityDMSO (100 mM) or Ethanol (100 mM)
Storage Protect from light
+2°C to +8°C
Do Not Freeze Ok to freeze
Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
Toxicity Standard Handling
ReferencesAdams, C. et al., 2007. CNS Drug Rev. 13, 308.
Pin, J.P., et al., 2007. Curr. Neuropharmacol. 5, 195.