Millipore Sigma Vibrant Logo
Attention: We have moved. Merck Millipore products are no longer available for purchase on MerckMillipore.com.Learn More

539684 PKA Inhibitor 6-22 Amide - CAS 121932-06-7 - Calbiochem

539684
  
Purchase on Sigma-Aldrich

Přehled

Tabulka spec. kláve

CAS #Empirical Formula
121932-06-7C₈₀H₁₃₀N₂₈O₂₄
Description
OverviewA potent and competitive inhibitor of protein kinase A (Ki = 1.7 nM).
Catalogue Number539684
Brand Family Calbiochem®
SynonymsPKI 6-22 Amide, TYADFIASGRTGRRNAI-NH₂, Protein Kinase A Inhibitor 6-22 Amide, PKA Inhibitor VIII
References
ReferencesGlass, D.B., et al. 1989. J. Biol. Chem. 264, 8802.
Kemp, B.E., et al. 1988. Methods Enzymol. 159, 173.
Product Information
CAS number121932-06-7
ATP CompetitiveN
FormSolid
FormulationSupplied as a trifluoroacetate salt.
Hill FormulaC₈₀H₁₃₀N₂₈O₂₄
Chemical formulaC₈₀H₁₃₀N₂₈O₂₄
Hygroscopic Hygroscopic
ReversibleN
Sold on the basis of peptide contentY
Quality LevelMQ100
Biological Information
Primary TargetPKA
Primary Target K<sub>i</sub> 1.7 nM against protein kinase A
Purity≥97% by HPLC
Physicochemical Information
Cell permeableN
Peptide ContentY
Peptide SequenceH-Thr-Tyr-Ala-Asp-Phe-Ile-Ala-Ser-Gly-Arg-Thr-Gly-Arg-Arg-Asn-Ala-Ile-NH₂
Storage and Shipping Information
Ship Code Ambient Temperature Only
Toxicity Standard Handling
Storage -20°C
Hygroscopic Hygroscopic
Do not freeze Ok to freeze
Special InstructionsFollowing initial thaw, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
Global Trade Item Number
Katalogové číslo GTIN
539684 0