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420305 K-252c - CAS 85753-43-1 - Calbiochem

420305
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Overview

Key Spec Table

CAS #Empirical Formula
85753-43-1C₂₀H₁₃N₃O

Products

Catalogue NumberPackaging Qty/Pack
420305-1MG Plastic ampoule 1 mg
Description
OverviewA cell-permeable, reversible, and ATP-competitive inhibitor of protein kinase C (IC50 = 2.45 µM) and protein kinase A (IC50 = 25.7 µM).
Catalogue Number420305
Brand Family Calbiochem®
References
ReferencesFabre, S., et al. 1993. Bioorg. Med. Chem. 1, 193.
Nakanishi, S., et al. 1986. J. Antibiot. 39, 1066.
Product Information
CAS number85753-43-1
ATP CompetitiveY
FormOff-white solid
Hill FormulaC₂₀H₁₃N₃O
Chemical formulaC₂₀H₁₃N₃O
ReversibleY
Structure formula ImageStructure formula Image
Quality LevelMQ100
Biological Information
Primary TargetPKC
Primary Target IC<sub>50</sub>2.45 µM against protein kinase C
Purity≥95% by HPLC
Physicochemical Information
Cell permeableY
Storage and Shipping Information
Ship Code Ambient Temperature Only
Toxicity Standard Handling
Storage +2°C to +8°C
Do not freeze Ok to freeze
Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C.
Global Trade Item Number
Catalogue Number GTIN
420305-1MG 04055977210927