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539746 InhibitorSelect™ 96-Well Protein Kinase Inhibitor Library III - Calbiochem

The InhibitorSelect™ 96-Well Protein Kinase Inhibitor Library III controls the biological activity of InhibitorSelect™. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

MSDS (material safety data sheet) or SDS, CoA and CoQ, dossiers, brochures and other available documents.
539746
  
Purchase on Sigma-Aldrich

Overview

Replacement Information
Description
Overview

This product has been discontinued.



The InhibitorSelect™ 96-Well Protein Kinase Inhibitor Library III consists of 84, well-characterized protein kinase inhibitors, the majority of which are cell-permeable and ATP-competitive. This serine/threonine-selective library will be useful for target identification in drug discovery, biochemical pathway analysis, screening new protein kinases, and other pharmaceutical-related applications.
Supplied with a CD containing comprehensive documentation for each inhibitor. Please contact technical service for further details.

Download a list of all inhibitors of library III, including a comprehensive data set.
Catalogue Number539746
Brand Family Calbiochem®
Application Data

** Total higher than 84, as some inhibitors target kinases in other branches as well AGC: PKA, PKG, and PKC Containing Group TKL: Tyrosine Kinase-Like Group CMGC: Cdk, MAP, GSK-3, and CLK Containing Group CAMK: Ca2+/Calmodulin Dependent Protein Kinases STE: Yeast Sterile Protein Kinases TK: Tyrosine Kinase
References
Product Information
Form96-well plate
Formulation81 inhibitors are supplied at a concentration of 10 mM and 3 inhibitors are supplied at a concentration of 5 mM in DMSO (50 µl/well).
Hygroscopic Hygroscopic
Applications
Biological Information
Physicochemical Information
Dimensions
Materials Information
Toxicological Information
Safety Information according to GHS
Safety Information
R PhraseR: 36/38

Irritating to eyes and skin.
S PhraseS: 26

In case of contact with eyes, rinse immediately with plenty of water and seek medical advice.
Product Usage Statements
Storage and Shipping Information
Ship Code Dry Ice Only
Toxicity Irritant
Storage ≤ -70°C
Protect from Light Protect from light
Hygroscopic Hygroscopic
Avoid freeze/thaw Avoid freeze/thaw
Do not freeze Ok to freeze
Special InstructionsThe contents of this pouch have been purged under nitrogen and are vacuum sealed. Cut open the pouch, take the plate out of the pouch, and let it thaw at room temperature. Please remove the lid gently. To re-store, purge with an inert gas, replace the lid tightly, place in a sealable bag, and store at -70°C in an upright position. Minimize freeze/thaw cycles. This product is stable for one year after receipt.
Packaging Information
Packaged under inert gas Packaged under inert gas
Transport Information
Supplemental Information
Specifications
Global Trade Item Number
Catalogue Number GTIN
539746 0

Documentation

InhibitorSelect™ 96-Well Protein Kinase Inhibitor Library III - Calbiochem SDS

Title

Safety Data Sheet (SDS) 

InhibitorSelect™ 96-Well Protein Kinase Inhibitor Library III - Calbiochem Certificates of Analysis

TitleLot Number
539746

Data Sheet

Title
Reprogramming Cell Fate and Function Novel Strategies for iPSC Generation, Characterization, and Differentiation

Citations

Title
  • Hou, P., et al. 2013. Science 341, 651.
  • Ali, H.A., et al. 2013. ACS Chem. Biol. in press.
  • Zhonghan Li1 and Tariq M. Ranal. 2012. Nature Comm. 3, 1085.
  • Cohen, T., et al. 2012. Biochem. J. in press.
  • Elkaim, J., 2012. Biochem. J. in press.
  • Baxter, B.K., et al. 2011. ACS Chem. Biol. in press.
  • Wong, S.W., et al. 2010. Breast Cancer Res. Treat. in press.
  • Chou, T-F. and Deshaies, R.J., 2011. JBC Papers in Press.
  • Gronenberg, L.S., and Kahne, d., 2009. J. AM. CHEM. SOC. 10.1021/ja910361r
    		•
    Data Sheet

    Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

    Revision11-September-2012 JSW
    Application Data

    ** Total higher than 84, as some inhibitors target kinases in other branches as well AGC: PKA, PKG, and PKC Containing Group TKL: Tyrosine Kinase-Like Group CMGC: Cdk, MAP, GSK-3, and CLK Containing Group CAMK: Ca2+/Calmodulin Dependent Protein Kinases STE: Yeast Sterile Protein Kinases TK: Tyrosine Kinase
    DescriptionThe InhibitorSelect™ 96-Well Protein Kinase Inhibitor Library III consists of 84 well-characterized protein kinase inhibitors, the majority of which are cell-permeable and ATP-competitive. This serine/threonine-selective library is useful for target identification in drug discovery, biochemical pathway analysis, screening new protein kinases, and other pharmaceutical-related applications. Supplied with a CD containing comprehensive documentation for each inhibitor. Please contact technical service for further details.
    Form96-well plate
    Formulation81 inhibitors are supplied at a concentration of 10 mM and 3 inhibitors are supplied at a concentration of 5 mM in DMSO (50 µl/well).
    Intert gas (Yes/No) Packaged under inert gas
    Storage Protect from light
    Avoid freeze/thaw
    ≤ -70°C
    Hygroscopic
    Do Not Freeze Ok to freeze
    Special InstructionsThe contents of this pouch have been purged under nitrogen and are vacuum sealed. Cut open the pouch, take the plate out of the pouch, and let it thaw at room temperature. Please remove the lid gently. To re-store, purge with an inert gas, replace the lid tightly, place in a sealable bag, and store at -70°C in an upright position. Minimize freeze/thaw cycles. This product is stable for one year after receipt.
    Toxicity Irritant
    Citation
  • Hou, P., et al. 2013. Science 341, 651.
  • Ali, H.A., et al. 2013. ACS Chem. Biol. in press.
  • Zhonghan Li1 and Tariq M. Ranal. 2012. Nature Comm. 3, 1085.
  • Cohen, T., et al. 2012. Biochem. J. in press.
  • Elkaim, J., 2012. Biochem. J. in press.
  • Baxter, B.K., et al. 2011. ACS Chem. Biol. in press.
  • Wong, S.W., et al. 2010. Breast Cancer Res. Treat. in press.
  • Chou, T-F. and Deshaies, R.J., 2011. JBC Papers in Press.
  • Gronenberg, L.S., and Kahne, d., 2009. J. AM. CHEM. SOC. 10.1021/ja910361r
    		•