203292 Sigma-AldrichBisindolylmaleimide II - CAS 137592-45-1 - Calbiochem
A potent, cell permeable, reversible, ATP-competitive and selective inhibitor of protein kinase C (IC₅₀ = 13 nM).
More>> A potent, cell permeable, reversible, ATP-competitive and selective inhibitor of protein kinase C (IC₅₀ = 13 nM). Less<<Bisindolylmaleimide II - CAS 137592-45-1 - Calbiochem MSDS (material safety data sheet) or SDS, CoA and CoQ, dossiers, brochures and other available documents.
Synonyms: 2-[1-[2-(1-Methylpyrrolidino)ethyl]-1H-indol-3-yl]-3-(1H-indol-3-yl)maleimide
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Overview
Key Spec Table
| CAS # | Empirical Formula |
|---|---|
| 137592-45-1 | C₂₇H₂₆N₄O₂ |
| References | |
|---|---|
| References | Toullec, D., et al. 1991. J. Biol. Chem. 266, 15771. |
| Product Information | |
|---|---|
| CAS number | 137592-45-1 |
| ATP Competitive | Y |
| Form | Orange solid |
| Hill Formula | C₂₇H₂₆N₄O₂ |
| Chemical formula | C₂₇H₂₆N₄O₂ |
| Reversible | Y |
| Structure formula Image | |
| Biological Information | |
|---|---|
| Primary Target | PKC |
| Primary Target IC<sub>50</sub> | 13 nM against protein kinase C |
| Purity | ≥95% by HPLC |
| Physicochemical Information | |
|---|---|
| Cell permeable | Y |
| Global Trade Item Number | |
|---|---|
| Catalogue Number | GTIN |
| 203292 | 0 |