Millipore Sigma Vibrant Logo
Attention: We have moved. Merck Millipore products are no longer available for purchase on MerckMillipore.com.Learn More

182200 βARK1 Inhibitor - CAS 24269-96-3 - Calbiochem

182200
Purchase on Sigma-Aldrich

Áttekintés

Kulcsspecifikációk táblázata

CAS #Empirical Formula
24269-96-3C₁₂H₉NO₆

Products

KatalógusszámCsomagolás Menny./csomag
182200-5MG Muanyagampulla 5 mg
Description
OverviewA selective inhibitor of βARK1 (β-Adrenergic Receptor Kinase 1) (IC50 = 126 µM). Has no inhibitory activity against protein kinase A (PKA).
Catalogue Number182200
Brand Family Calbiochem®
Synonymsβ-Adrenergic Receptor Kinase1 Inhibitor, GRK2 Inhibitor, Methyl 5-[2-(5-nitro-2-furyl)vinyl]-2-furoate
References
ReferencesIino, M., et al. 2002. J. Med. Chem. 45, 2150.
Product Information
CAS number24269-96-3
ATP CompetitiveN
FormYellow to orange solid
Hill FormulaC₁₂H₉NO₆
Chemical formulaC₁₂H₉NO₆
ReversibleN
Structure formula ImageStructure formula Image
Quality LevelMQ100
Biological Information
Primary TargetβARK1 (β-Adrenergic Receptor Kinase 1)
Primary Target IC<sub>50</sub>126 µM against βARK1 (β-Adrenergic Receptor Kinase 1)
Purity≥97% by HPLC
Physicochemical Information
Cell permeableN
Storage and Shipping Information
Ship Code Ambient Temperature Only
Toxicity Standard Handling
Storage -20°C
Protect from Light Protect from light
Do not freeze Ok to freeze
Special InstructionsFollowing reconstitution aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C.
Packaging Information
Packaged under inert gas Packaged under inert gas
Global Trade Item Number
Katalógusszám GTIN
182200-5MG 04055977205046