Custom Premix Selecting "Custom Premix" option means that all of the beads you have chosen will be premixed in manufacturing before the kit is sent to you.
A highly potent and selective non-alkaloid positive allosteric modulator of Κ-opioid receptors (Ki = 4.3 nM and 16 nM for native and cloned κ-opioid receptors, respectively). Also acts as a D2DR partial agonist (Ki = 5-10 nM). Used in studies of addition.
Catalogue Number
508159
Brand Family
Calbiochem®
Synonyms
κ-opioid Receptor Agonist, Salvinorin A, Divinorin A
References
References
Roth, B. et al., 2002. PNAS.99, 11934. Valdés III., j., et al., 1984. J. Organic Chem.49, 4716. Ortega, A., et al., 1982. J. of Chem. Society, Perkins Transactions I. 2505.
Roth, B. et al., 2002. PNAS.99, 11934. Valdés III., j., et al., 1984. J. Organic Chem.49, 4716. Ortega, A., et al., 1982. J. of Chem. Society, Perkins Transactions I. 2505.
数据表
Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.
Revision
31-October-2013 JSW
Synonyms
κ-opioid Receptor Agonist, Salvinorin A, Divinorin A
Description
A highly potent and selective non-alkaloid positive allosteric modulator of Κ-opioid receptors (Ki = 4.3 nM and 16 nM for native and cloned κ-opioid receptors, respectively). Also acts as a D2DR partial agonist (Ki = 5-10 nM). Used in studies of addition.
Form
White solid
CAS number
83729-01-5
Chemical formula
C₂₃H₂₈O₈
Structure formula
Purity
≥98% by HPLC
Solubility
DMSO (50 mM) or Ethanol (10 mM)
Storage
Protect from light
≤ -70°C
Do Not Freeze
Ok to freeze
Special Instructions
Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
Toxicity
Standard Handling
References
Roth, B. et al., 2002. PNAS.99, 11934. Valdés III., j., et al., 1984. J. Organic Chem.49, 4716. Ortega, A., et al., 1982. J. of Chem. Society, Perkins Transactions I. 2505.
