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539610 PKCζ/ι Pseudosubstrate Inhibitor - Calbiochem

The PKCζ/ι Pseudosubstrate Inhibitor controls the biological activity of PKCζ/ι. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

MSDS (material safety data sheet) or SDS, CoA and CoQ, dossiers, brochures and other available documents.

Synonyms: SIYRRGARRWRKL, Protein Kinase Cζ/ι Pseudosubstrate Inhibitor

Primary Target: PKCζ
539610
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Overview

Key Spec Table

Empirical Formula
C₇₆H₁₂₈N₃₀O₁₆

Products

Catalogue NumberPackaging Qty/Pack
539610-500UG Plastic ampoule 500 μg
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Description
OverviewA selective, reversible, and substrate competitive inhibitor of protein kinase Cζ and protein kinase Cι (PKCζ/ι) isozymes.
Catalogue Number539610
Brand Family Calbiochem®
SynonymsSIYRRGARRWRKL, Protein Kinase Cζ/ι Pseudosubstrate Inhibitor
References
ReferencesSajan, M.P., et al. 1999. J. Biol. Chem. 274, 30495.
Laudanna, C., et al. 1998. J. Biol. Chem. 273, 30306.
Standaert, M.L., et al. 1997. J. Biol. Chem. 272, 30075.
Product Information
ATP CompetitiveN
FormLyophilized
FormulationSupplied as a trifluoroacetate salt.
Hill FormulaC₇₆H₁₂₈N₃₀O₁₆
Chemical formulaC₇₆H₁₂₈N₃₀O₁₆
Hygroscopic Hygroscopic
ReversibleY
Quality LevelMQ100
Biological Information
Primary TargetPKCζ
Purity≥95% by HPLC
Physicochemical Information
Cell permeableN
Peptide SequenceH-Ser-Ile-Tyr-Arg-Arg-Gly-Ala-Arg-Arg-Trp-Arg-Lys-Leu-OH
Storage and Shipping Information
Ship Code Ambient Temperature Only
Toxicity Standard Handling
Storage -20°C
Hygroscopic Hygroscopic
Do not freeze Ok to freeze
Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
Global Trade Item Number
Catalogue Number GTIN
539610-500UG 04055977194777