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05-22-3838 BQ-788, Sodium Salt - CAS - Calbiochem

BQ-788, Sodium Salt - CAS - Calbiochem MSDS (material safety data sheet) or SDS, CoA and CoQ, dossiers, brochures and other available documents.

Synonyms: N-cis-2,6-Dimethylpiperidinocarbonyl-L-γ-MeLeu-D-Trp(MeOCO)-D-Nle-OH, Na

Primary Target: ETB-receptor antagonist
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05-22-3838
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Overview

Replacement Information

Key Spec Table

Empirical Formula
C₃₄H₅₀N₅O₇Na

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      Description
      OverviewHighly selective ETB-receptor antagonist (IC50 = 1.2 nM).
      Catalogue Number05-22-3838
      Brand Family Calbiochem®
      SynonymsN-cis-2,6-Dimethylpiperidinocarbonyl-L-γ-MeLeu-D-Trp(MeOCO)-D-Nle-OH, Na
      References
      ReferencesOkada, M., and Nishikibe, M. 2002. Cardiovasc. Drug Reviews 20, 53.
      Taniai, H., et al. 2001. Hepatology 33, 894.
      Fukuroda, T., et al. 1994. Biochem. Biophys. Res. Commun. 199, 1461.
      Ishikawa, K., et al. 1994. Proc. Natl. Acad. Sci. USA 91, 4892.
      Product Information
      ATP CompetitiveN
      FormWhite to off-white lyophilized solid
      Hill FormulaC₃₄H₅₀N₅O₇Na
      Chemical formulaC₃₄H₅₀N₅O₇Na
      ReversibleN
      Structure formula ImageStructure formula Image
      Quality LevelMQ100
      Applications
      Biological Information
      Primary TargetETB-receptor antagonist
      Primary Target IC<sub>50</sub>1.2 nM as ETB-receptor antagonist
      Purity≥95% by HPLC
      Physicochemical Information
      Cell permeableN
      Dimensions
      Materials Information
      Toxicological Information
      Safety Information according to GHS
      Safety Information
      Product Usage Statements
      Storage and Shipping Information
      Ship Code Ambient Temperature Only
      Toxicity Standard Handling
      Storage -20°C
      Protect from Moisture Protect from moisture
      Do not freeze Ok to freeze
      Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). DMSO and Methano:H₂O stock solutions are stable for up to 2 months at -20°C.
      Packaging Information
      Transport Information
      Supplemental Information
      Specifications
      Global Trade Item Number
      Catalogue Number GTIN
      05-22-3838-1MG 04055977225051

      Documentation

      BQ-788, Sodium Salt - CAS - Calbiochem SDS

      Title

      Safety Data Sheet (SDS) 

      BQ-788, Sodium Salt - CAS - Calbiochem Certificates of Analysis

      TitleLot Number
      05-22-3838

      References

      Reference overview
      Okada, M., and Nishikibe, M. 2002. Cardiovasc. Drug Reviews 20, 53.
      Taniai, H., et al. 2001. Hepatology 33, 894.
      Fukuroda, T., et al. 1994. Biochem. Biophys. Res. Commun. 199, 1461.
      Ishikawa, K., et al. 1994. Proc. Natl. Acad. Sci. USA 91, 4892.
      Data Sheet

      Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

      Revision18-September-2008 RFH
      SynonymsN-cis-2,6-Dimethylpiperidinocarbonyl-L-γ-MeLeu-D-Trp(MeOCO)-D-Nle-OH, Na
      DescriptionA highly selective and competitive ETB receptor antagonist (IC50 = 1.2 nM).
      FormWhite to off-white lyophilized solid
      Chemical formulaC₃₄H₅₀N₅O₇Na
      Structure formulaStructure formula
      Purity≥95% by HPLC
      SolubilityDMSO (2 mg/ml), Methanol:H₂O (3:1) (2 mg/ml), or 0.01% NH₄OH (1 mg/ml)
      Storage Protect from moisture
      -20°C
      Do Not Freeze Ok to freeze
      Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). DMSO and Methano:H₂O stock solutions are stable for up to 2 months at -20°C.
      Toxicity Standard Handling
      ReferencesOkada, M., and Nishikibe, M. 2002. Cardiovasc. Drug Reviews 20, 53.
      Taniai, H., et al. 2001. Hepatology 33, 894.
      Fukuroda, T., et al. 1994. Biochem. Biophys. Res. Commun. 199, 1461.
      Ishikawa, K., et al. 1994. Proc. Natl. Acad. Sci. USA 91, 4892.