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361555 GSK-3 Inhibitor XIII - CAS 404828-08-6 - Calbiochem

The GSK-3 Inhibitor XIII, also referenced under CAS 404828-08-6, controls the biological activity of GSK-3. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

FDS (Fiches de données de sécurité), certificats d’analyse (CoA) et de qualité (CoQ), dossiers, brochures et autres documents disponibles.

Synonymes: (5-Methyl-1H-pyrazol-3-yl)-(2-phenylquinazolin-4-yl)amine

Primary Target: GSK-3
361555
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Aperçu

Replacement Information

Tableau de caractéristiques principal

CAS #Empirical Formula
404828-08-6C₁₈H₁₅N₅

Products

RéférenceConditionnement Qté
361555-1MG Ampoule plast. 1 mg
361555-5MG Ampoule plast. 5 mg
Description
OverviewAn aminopyrazole compound that acts as a potent and ATP-binding site inhibitor of GSK-3 with a Ki of 24 nM.
Catalogue Number361555
Brand Family Calbiochem®
Synonyms(5-Methyl-1H-pyrazol-3-yl)-(2-phenylquinazolin-4-yl)amine
References
ReferencesPierce, A.C., et al. 2005. J. Med. Chem. 48, 1278.
Product Information
CAS number404828-08-6
ATP CompetitiveN
FormWhite solid
Hill FormulaC₁₈H₁₅N₅
Chemical formulaC₁₈H₁₅N₅
ReversibleN
Structure formula ImageStructure formula Image
Quality LevelMQ100
Applications
Biological Information
Primary TargetGSK-3
Primary Target K<sub>i</sub>24 nM against GSK-3
Purity≥95% by HPLC
Physicochemical Information
Cell permeableN
Dimensions
Materials Information
Toxicological Information
Safety Information according to GHS
Safety Information
Product Usage Statements
Storage and Shipping Information
Ship Code Ambient Temperature Only
Toxicity Carcinogenic / Teratogenic
Storage +2°C to +8°C
Protect from Light Protect from light
Do not freeze Ok to freeze
Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C.
Packaging Information
Transport Information
Supplemental Information
Specifications
Global Trade Item Number
Référence GTIN
361555-1MG 04055977214147
361555-5MG 04055977214154

Documentation

GSK-3 Inhibitor XIII - CAS 404828-08-6 - Calbiochem FDS

Titre

Fiche de données de sécurité des matériaux (FDS) 

GSK-3 Inhibitor XIII - CAS 404828-08-6 - Calbiochem Certificats d'analyse

TitreNuméro de lot
361555

Références bibliographiques

Aperçu de la référence bibliographique
Pierce, A.C., et al. 2005. J. Med. Chem. 48, 1278.
Fiche technique

Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

Revision01-July-2008 RFH
Synonyms(5-Methyl-1H-pyrazol-3-yl)-(2-phenylquinazolin-4-yl)amine
DescriptionA potent and ATP-competitive inhibitor of GSK-3 (Ki = 24 nM).
FormWhite solid
CAS number404828-08-6
Chemical formulaC₁₈H₁₅N₅
Structure formulaStructure formula
Purity≥95% by HPLC
SolubilityDMSO (5 mg/ml)
Storage Protect from light
+2°C to +8°C
Do Not Freeze Ok to freeze
Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C.
Toxicity Carcinogenic / Teratogenic
ReferencesPierce, A.C., et al. 2005. J. Med. Chem. 48, 1278.