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371725 GPR43 (FFA2) Agonist - CAS 1208552-99-1 - Calbiochem

GPR43 (FFA2) Agonist is an allosteric agonist of FFA2 (GPR43). Displays a left-shifted acetate dose response (IC50 = 0.7 µM) & 111% efficacy relative to acetate in hFFA2 forskolin-induced cAMP assays.

FDS (Fiches de données de sécurité), certificats d’analyse (CoA) et de qualité (CoQ), dossiers, brochures et autres documents disponibles.

Synonymes: (S)-2-(4-chlorophenyl)-3,3-dimethyl-N-(5-phenylthiazol-2-yl)butanamide

371725
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Aperçu

Replacement Information

Tableau de caractéristiques principal

CAS #Empirical Formula
1208552-99-1C₂₁H₂₁ClN₂OS

Products

RéférenceConditionnement Qté
371725-10MG Flacon en verre 10 mg
Description
OverviewA phenylacetamide compound that acts as an allosteric agonist of FFA2 (GPR43), demonstrating a left-shifted acetate dose response (IC50 = 0.7 µM) and 111% efficacy relative to acetate in hFFA2 forskolin-induced cAMP assays.
Catalogue Number371725
Brand Family Calbiochem®
Synonyms(S)-2-(4-chlorophenyl)-3,3-dimethyl-N-(5-phenylthiazol-2-yl)butanamide
References
ReferencesWang, Y., et al. 2009. Bioorg. Med. Chem. Lett. 20, 493.
Product Information
CAS number1208552-99-1
FormWhite solid
Hill FormulaC₂₁H₂₁ClN₂OS
Chemical formulaC₂₁H₂₁ClN₂OS
Structure formula ImageStructure formula Image
Quality LevelMQ100
Applications
ApplicationGPR43 (FFA2) Agonist is an allosteric agonist of FFA2 (GPR43). Displays a left-shifted acetate dose response (IC50 = 0.7 µM) & 111% efficacy relative to acetate in hFFA2 forskolin-induced cAMP assays.
Biological Information
Purity>98% by HPLC
Physicochemical Information
Dimensions
Materials Information
Toxicological Information
Safety Information according to GHS
Safety Information
Product Usage Statements
Storage and Shipping Information
Ship Code Ambient Temperature Only
Toxicity Standard Handling
Storage +2°C to +8°C
Do not freeze Ok to freeze
Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
Packaging Information
Transport Information
Supplemental Information
Specifications
Global Trade Item Number
Référence GTIN
371725-10MG 04055977213270

Documentation

GPR43 (FFA2) Agonist - CAS 1208552-99-1 - Calbiochem FDS

Titre

Fiche de données de sécurité des matériaux (FDS) 

GPR43 (FFA2) Agonist - CAS 1208552-99-1 - Calbiochem Certificats d'analyse

TitreNuméro de lot
371725

Références bibliographiques

Aperçu de la référence bibliographique
Wang, Y., et al. 2009. Bioorg. Med. Chem. Lett. 20, 493.
Fiche technique

Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

Revision06-June-2015 JSW
Synonyms(S)-2-(4-chlorophenyl)-3,3-dimethyl-N-(5-phenylthiazol-2-yl)butanamide
DescriptionA phenylacetamide compound that acts as an allosteric agonist of FFA2 (GPR43), demonstrating a left-shifted acetate dose response (IC50 = 0.7 µM) and 111% efficacy relative to acetate in hFFA2 forskolin-induced cAMP assays.
FormWhite solid
CAS number1208552-99-1
Chemical formulaC₂₁H₂₁ClN₂OS
Structure formulaStructure formula
Purity>98% by HPLC
SolubilityDMSO (50 mg/ml)
Storage +2°C to +8°C
Do Not Freeze Ok to freeze
Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
Toxicity Standard Handling
ReferencesWang, Y., et al. 2009. Bioorg. Med. Chem. Lett. 20, 493.