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211280 Capsazepine - CAS 138977-28-3 - Calbiochem

211280
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Overview

Key Spec Table

CAS #Empirical Formula
138977-28-3C₁₉H₂₁N₂O₂SCl

Products

Catalogue NumberPackaging Qty/Pack
211280-10MG Plastic ampoule 10 mg
Description
OverviewA competitive antagonist of Capsaicin (Cat. No. 211274) and resiniferatoxin. Capsazepine (1 µM) blocks capsaicin (60 nM) stimulated firing of C-fibers.
Catalogue Number211280
Brand Family Calbiochem®
SynonymsN-[2-(4-Chlorophenyl)ethyl]-1,3,4,5-tetrahydro-7,8-dihydroxy-2H-2-benzazepine-2-carbothioamide
References
ReferencesFox, A.J., et al. 1995. Neuroscience 67, 741.
Ellis, J.L., and Undem, B.J. 1994. J. Pharmacol. Exp. Ther. 268, 85.
Walpole, C.S.J., et al. 1994. J. Med. Chem. 37, 1942.
Szallasi, A., et al. 1993. J. Pharmacol. Exp. Therap. 267, 728.
Product Information
CAS number138977-28-3
ATP CompetitiveN
FormOff-white solid
Hill FormulaC₁₉H₂₁N₂O₂SCl
Chemical formulaC₁₉H₂₁N₂O₂SCl
ReversibleN
Structure formula ImageStructure formula Image
Quality LevelMQ100
Biological Information
Primary TargetA competitive antagonist of Capsaicin and resiniferatoxin
Purity≥97% by HPLC
Physicochemical Information
Cell permeableN
Storage and Shipping Information
Ship Code Ambient Temperature Only
Toxicity Standard Handling
Storage +15°C to +30°C
Do not freeze Ok to freeze
Special InstructionsUnstable in solution; reconstitute just prior to use.
Global Trade Item Number
Catalogue Number GTIN
211280-10MG 04055977219180