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505986 SR95531 (Gabazine) - CAS 104104-50-9 - Calbiochem

Overview

Key Spec Table

CAS #Empirical Formula
104104-50-9C₁₅H₁₇N₃O₃•HBr

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5.05986.0001
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      Glass bottle 10 mg
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      Description
      OverviewA selective, competitive antagonist of GABAA receptor (IC50 = 440 nM) that does not affect pentobarbitone or etomidate- induced currents even at high concentrations (~100 µM). Also shown to block glycine receptors, but with low affinity (Kb = 190 µM).
      Catalogue Number505986
      Brand Family Calbiochem®
      SynonymsGABAA Receptor Antagonist, SR-95531, Gabazine, SR95531, SR 95531
      References
      ReferencesMuroi, Y., et al. 2009. Biophys. J. 96, 499.
      Beato, M., et al. 2007. J. Physiol. 580, 171.
      Uchida, I., et al. 1996. Eur. J. Pharmacol. 307, 89.
      Product Information
      CAS number104104-50-9
      FormWhite solid
      Hill FormulaC₁₅H₁₇N₃O₃•HBr
      Chemical formulaC₁₅H₁₇N₃O₃•HBr
      Structure formula ImageStructure formula Image
      Quality LevelMQ100
      Biological Information
      Primary TargetGABAA
      Primary Target IC<sub>50</sub>440 nM
      Purity≥98% by HPLC
      Storage and Shipping Information
      Ship Code Shipped at Ambient Temperature or with Blue Ice or with Dry Ice
      Toxicity Standard Handling
      Storage +2°C to +8°C
      Protect from Light Protect from light
      Do not freeze Ok to freeze
      Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
      Global Trade Item Number
      Catalogue Number GTIN
      5.05986.0001 04055977262582