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182200 βARK1 Inhibitor - CAS 24269-96-3 - Calbiochem

Overview

Key Spec Table

CAS #Empirical Formula
24269-96-3C₁₂H₉NO₆

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182200-5MG
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      Description
      OverviewA selective inhibitor of βARK1 (β-Adrenergic Receptor Kinase 1) (IC50 = 126 µM). Has no inhibitory activity against protein kinase A (PKA).
      Catalogue Number182200
      Brand Family Calbiochem®
      Synonymsβ-Adrenergic Receptor Kinase1 Inhibitor, GRK2 Inhibitor, Methyl 5-[2-(5-nitro-2-furyl)vinyl]-2-furoate
      References
      ReferencesIino, M., et al. 2002. J. Med. Chem. 45, 2150.
      Product Information
      CAS number24269-96-3
      ATP CompetitiveN
      FormYellow to orange solid
      Hill FormulaC₁₂H₉NO₆
      Chemical formulaC₁₂H₉NO₆
      ReversibleN
      Structure formula ImageStructure formula Image
      Quality LevelMQ100
      Biological Information
      Primary TargetβARK1 (β-Adrenergic Receptor Kinase 1)
      Primary Target IC<sub>50</sub>126 µM against βARK1 (β-Adrenergic Receptor Kinase 1)
      Purity≥97% by HPLC
      Physicochemical Information
      Cell permeableN
      Storage and Shipping Information
      Ship Code Ambient Temperature Only
      Toxicity Standard Handling
      Storage -20°C
      Protect from Light Protect from light
      Do not freeze Ok to freeze
      Special InstructionsFollowing reconstitution aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C.
      Packaging Information
      Packaged under inert gas Packaged under inert gas
      Global Trade Item Number
      Catalogue Number GTIN
      182200-5MG 04055977205046